Beilstein J. Org. Chem.2019,15, 780–788, doi:10.3762/bjoc.15.74
derivatives showed antagonistic activity lacking isomer specificity.
Keywords: azobenzene; 5-HT3R; ioncurrents; photopharmacology; serotonin; Introduction
5-Hydroxytryptamine (5-HT), commonly known as serotonin [1][2] or enteramine [3][4], is a monoamine neurotransmitter and hormone which is produced in
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Graphical Abstract
Scheme 1:
Approach of the direct azologization of reported [60,61] serotonin 5-HT3R antagonists via replacement of a...